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產(chan)品名稱:TH 1020 1841460-82-9
規(gui)格(ge):10 mg、50 mg
貨(huo)號:GOY-01Y64882
Cas No.: 1841460-82-9
別(bie)名: N/A
化(hua)學名: N/A
分(fen)子(zi)式(shi): C23H15N7S2

分(fen)子(zi)量(liang): 453.54
溶(rong)解(jie)度: Chloroform: 1 mg/ml
儲存條(tiao)件: Store at -20°C
General tips For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping Condition Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chan)品說明:
Toll-like receptor (TLR) 5/Flagellin complex antagonist (IC50 = 0.85 μM). Competes with flagellin for TLR5 binding to inhibit the TLR5:flagellin interaction and subsequent downstream TNF-α secretion.Yan et al (2016) Pyrimidine triazole thioether derivatives as toll-like receptor 5 (TLR5)/flagellin complex inhibitors. Chem.Med.Chem. 11 822 PMID:26634412
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